Elagolix sodium (NBI-56418 sodium) [CAS 832720-36-2] - ChemeGen-活性小分子-抑制剂-激动剂

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Elagolix sodium (NBI-56418 sodium) [CAS 832720-36-2]

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产品详情

Cat. No.：	C105244	Chinese Name：	恶拉戈利钠盐
CAS：	832720-36-2	Formula：	C32H29F5N3NaO5
MWt：	653.57	Purity：	>98%
Solubility：	DMSO	Storage：	Powder -20°C 3 years; 4°C 2 years In solvent -80°C 6 months; -20°C 1 month
Research Area：	Endocrinology	Target：	GNRH Receptor
Description：	Elagolix sodium is a human GnRH receptor (GnRHR) antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.

[1]. Kim SM, et al. Discovery of an Orally Bioavailable Gonadotropin-Releasing Hormone Receptor Antagonist. J Med Chem. 2016 Oct 13;59(19):9150-9172. Epub 2016 Sep 27.

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